PF-06291874 - Powerful and Selective Glucagon Receptor Antagonist

REF #: 3199373
Procurenet
Short description

PF-06291874 is a powerful and selective glucagon receptor antagonist. It is an orally active compound, making it convenient for administration. The composition of PF-06291874 is as follows:

  • Chemical Name: N-[4-[(1S)-1-[3,5-Dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy]butyl]benzoyl]-alanine
  • CAS Number: 1393124-08-7
  • Purity: 98% (HPLC)
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  • Procurenet Team Tshim Sha Tsui
    Hong Kong Hong Kong 3 years
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Description

PF-06291874 - Powerful and Selective Glucagon Receptor Antagonist

PF-06291874 is a powerful and selective glucagon receptor antagonist. It is an orally active compound, making it convenient for administration.

Chemical Name

N-[4-[(1S)-1-[3,5-Dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy]butyl]benzoyl]-alanine

CAS Number

1393124-08-7

Purity

98% (HPLC)

Features

  • Powerful and selective glucagon receptor antagonist
  • Orally active compound, convenient for administration
  • High purity of 98% (HPLC)

Ingredients

PF-06291874 is composed of the following ingredients:

  • N-[4-[(1S)-1-[3,5-Dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy]butyl]benzoyl]-alanine: This chemical compound is the main active ingredient in PF-06291874. It acts as a powerful and selective glucagon receptor antagonist, blocking the glucagon receptor and inhibiting its effects. It is orally active, allowing for convenient administration.

Composition

The composition of PF-06291874 is carefully formulated to ensure its effectiveness as a glucagon receptor antagonist. The main components include:

  • 4-(trifluoromethyl)-1H-pyrazol-1-yl: This component is responsible for the pyrazol-1-yl structure of PF-06291874. It adds stability and structural integrity to the compound, allowing it to effectively bind to the glucagon receptor.
  • 3,5-Dimethyl: This component is a methyl group attached to the pyrazol-1-yl structure. It provides additional stability and contributes to the overall potency of PF-06291874.
  • Phenoxybutyl: This component is a phenoxy group attached to a butyl chain. It enhances the binding affinity of PF-06291874 to the glucagon receptor, making it a highly selective antagonist.
  • benzoyl-alanine: This component is a benzoyl group attached to an alanine residue. It further contributes to the selectivity and potency of PF-06291874 as a glucagon receptor antagonist.

These carefully selected components work together to create PF-06291874, a powerful and selective glucagon receptor antagonist.

Product Benefits

  • Powerful and selective: PF-06291874 is specifically designed to target and antagonize the glucagon receptor, effectively blocking its effects.
  • Convenient administration: Being orally active, PF-06291874 allows for easy and convenient administration.
  • High purity: With a purity level of 98% as measured by HPLC (High-Performance Liquid Chromatography), PF-06291874 ensures consistent quality and potency.

Applications

PF-06291874 has various applications in the field of pharmacology and drug research. Some of its potential applications include:

  • Treatment of metabolic disorders: Due to its glucagon receptor antagonist properties, PF-06291874 could be utilized in the development of therapeutic interventions for metabolic disorders such as diabetes and obesity.
  • Research tool: PF-06291874 can be used as a research tool to study the role of glucagon in various physiological processes and disease states.

Conclusion

PF-06291874 is a powerful and selective glucagon receptor antagonist that offers convenient oral administration and high purity. Its carefully designed composition ensures its effectiveness in blocking the glucagon receptor and inhibiting its effects. With its potential applications in the treatment of metabolic disorders and as a research tool, PF-06291874 is a valuable compound in the field of pharmacology and drug development.

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